Publications

Our scientific publications in high-quality journals reflect the quality of the innovative research in Entasis’ laboratories.

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Basarab GS, Brassil P, Doig P, Galullo V, Haimes HB, Kern G, Kutschke A, McNulty J, Schuck VJ, Stone G, and Gowravaram M

Novel DNA gyrase inhibiting spiropyrimidinetriones with a benzisoxazole scaffold: SAR and in vivo characterization

Journal of Medicinal Chemistry (2014)

Basarab GS, Galullo V, DeGrace N, Hauck S, Joubran C, and Wesolowski SS

Synthesis of a tetrahydronaphthyridine spiropyrimidinetrione DNA gyrase inhibiting antibacterial agent – differential substitution at all five carbon atoms of pyridine

Organic Letters (2014)